Laboratoire de Chimie de Coordination UPR 8241


Accueil

Jean-Luc STIGLIANI
MDC
0561333236
G173

Publications


2020

Fersing, C., Boudot, C., Castera-Ducros, C., Pinault, E., Hutter, S., Paoli-Lombardo, R., Primas, N., Pedron, J., Seguy, L., Bourgeade-Delmas, S., Sournia-Saquet, A., Stigliani, J. - L., Brossas, J. - Y., Paris, L., Valentin, A., Wyllie, S., Fairlamb, A. H., Boutet-Robinet, É., Corvaisier, S., Since, M., Malzert-Fréon, A., Destere, A., Mazier, D., Rathelot, P., Courtioux, B., Azas, N., Verhaeghe, P., & Vanelle, P. (2020). 8-Alkynyl-3-nitroimidazopyridines display potent antitrypanosomal activity against both T. b. brucei and cruzi. Eur. J. Med. Chem., 202, 112558/1–15.
Fersing, C., Boudot, C., Paoli-Lombardo, R., Primas, N., Pinault, E., Hutter, S., Castera-Ducros, C., Kabri, Y., Pedron, J., Bourgeade-Delmas, S., Sournia-Saquet, A., Stigliani, J. - L., Valentin, A., Azqueta, A., Muruzabal, D., Destere, A., Wyllie, S., Fairlamb, A. H., Corvaisier, S., Since, M., Malzert-Fréon, A., Di Giorgio, C., Rathelot, P., Azas, N., Courtioux, B., Vanelle, P., & Verhaeghe, P. (2020). Antikinetoplastid SAR study in 3-nitroimidazopyridine series: Identification of a novel non-genotoxic and potent anti-T. b. brucei hit-compound with improved pharmacokinetic properties. Eur. J. Med. Chem., 206, 112668/1–20.
Paludetto, M. - N., Stigliani, J. - L., Robert, A., Bernardes-Génisson, V., Chatelut, E., Puisset, F., & Arellano, C. (2020). Involvement of Pazopanib and Sunitinib aldehyde reactive metabolites in toxicity and drug–drug interactions in vitro and in patient samples. Chem. Res. Toxicol., 33(1), 181–190.
Pedron, J., Boudot, C., Brossas, J. - Y., Pinault, E., Bourgeade-Delmas, S., Sournia-Saquet, A., Boutet-Robinet, E., Destere, A., Tronnet, A., Bergé, J., Bonduelle, C., Deraeve, C., Pratviel, G., Stigliani, J. - L., Paris, L., Mazier, D., Corvaisier, S., Since, M., Malzert-Fréon, A., Wyllie, S., Milne, R., Fairlamb, A. H., Valentin, A., Courtioux, B., & Verhaeghe, P. (2020). New 8‑nitroquinolinone derivative displaying submicromolar in vitro activities against both Trypanosoma brucei and cruzi. ACS Med. Chem. Lett., 11, 464−472.
Reyser, T., To, T. H., Egwu, C., Paloque, L., Nguyen, M., Hamouy, A., Stigliani, J. - L., Bijani, C., Augereau, J. - M., Joly, J. - P., Portela, J., Havot, J., Marque, S. R. A., Boissier, J., Robert, A., Benoit-Vical, F., & Audran, G. (2020). Alkoxyamines designed as potential drugs against Plasmodium and Schistosoma parasites. Molecules, 25(17), 3838/1–23.

2019

Barakat, F., Vansteelandt, M., Triastuti, A., Jargeat, P., Jacquemin, D., Graton, J., Mejia, K., Cabanillas, B., Vendier, L., Stigliani, J. - L., Haddad, M., & Fabre, N. (2019). Thiodiketopiperazines with two spirocyclic centers extracted from Botryosphaeria mamane, an endophytic fungus isolated from Bixa orellana L. Phytochemistry, 158, 142–148.
Pipier, A., De Rache, A., Modeste, C., Amrane, S., Mothes-Martin, E., Stigliani, J. - L., Calsou, P., Mergny, J. - L., Pratviel, G., & Gomez, D. (2019). G-Quadruplex binding optimization by gold(iii) insertion into the center of a porphyrin. Dalton Trans., 48(18), 6091–6099.
Stigliani, J. - L., & Bernardes-Génisson, V. (2019). New insights into the chemical behavior of S-oxide derivatives of thiocarbonyl-containing antitubercular drugs and the influence on their mechanisms of action and toxicity. Ann. Pharm. Fr., 77(2), 126–135.

2018

Fersing, C., Boudot, C., Pedron, J., Hutter, S., Primas, N., Castera-Ducros, C., Bourgeade-Delmas, S., Sournia-Saquet, A., Moreau, A., Cohen, A., Stigliani, J. - L., Pratviel, G., Crozet, M. D., Wyllie, S., Fairlamb, A., Valentin, A., Rathelot, P., Azas, N., Courtioux, B., Verhaeghe, P., & Vanelle, P. (2018). 8-Aryl-6-chloro-3-nitro-2-(phenylsulfonylmethyl)imidazo[1,2-a]pyridines as potent antitrypanosomatid molecules bioactivated by type 1 nitroreductases. Eur. J. Med. Chem., 157, 115–126.
Nguyen, M., Stigliani, J. - L., Bijani, C., Verhaeghe, P., Pratviel, G., & Bonduelle, C. (2018). Ionic polypeptide polymers with unusual β-sheet stability. Biomacromolecules, 19(10), 4068–4074.